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2020
Prevalence and significance of the commonest phosphorylated motifs in the human proteome: a global analysis
Cellular and Molecular Life Sciences
2020
Discovery of a novel kinase hinge binder fragment by dynamic undocking
RSC Medicinal Chemistry
2020
Novel method to identify group-specific non-catalytic pockets of human kinome for drug design
RSC Advances
2020
KinomeRun: An interactive utility for kinome target screening and interaction fingerprint analysis towards holistic visualization on kinome tree
Chemical Biology & Drug Design
2020
Discovery of a Novel Dual-Target Inhibitor of ERK1 and ERK5 That Induces Regulated Cell Death to Overcome Compensatory Mechanism in Specific Tumor Types
Journal of Medicinal Chemistry
2020
Pyridin-2(1H)one derivatives: A possible new class of therapeutics for mechanical allodynia
European Journal of Medicinal Chemistry
2020
Evolution of new enzymes by gene duplication and divergence
The FEBS Journal
2019
Characterization of the Src-regulated kinome identifies SGK1 as a key mediator of Src-induced transformation
Nature Communications
2019
Investigation of Crystal Structures in Structure-Based Virtual Screening for Protein Kinase Inhibitors
Journal of Chemical Information and Modeling
2019
Methods in Molecular Biology
2019
HKPocket: human kinase pocket database for drug design
BMC Bioinformatics
2019
A Structurally-Validated Multiple Sequence Alignment of 497 Human Protein Kinase Domains
Scientific Reports
2019
CoralP: Flexible visualization of the human phosphatome
Journal of Open Source Software
2019
KinomeX: a web application for predicting kinome-wide polypharmacology effect of small molecules
Bioinformatics
2019
Regulated Phosphosignaling Associated with Breast Cancer Subtypes and Druggability
Molecular & Cellular Proteomics
2018
Exploring Selectivity of Multikinase Inhibitors across the Human Kinome
ACS Omega
2018
Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition
Bioorganic & Medicinal Chemistry
2018
Comprehensive assessment of nine docking programs on type II kinase inhibitors: prediction accuracy of sampling power, scoring power and screening power
Briefings in Bioinformatics
2018
Highly Selective, Potent, and Oral mTOR Inhibitor for Treatment of Cancer as Autophagy Inducer
Journal of Medicinal Chemistry
2018
Design, synthesis and evaluation of (R)-3-(7-(methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-5-azaspiro[2.4]heptan-5-yl)-3-oxopropanenitrile as a JAK1-selective inhibitor
MedChemComm
2018
Discovery of 4-ethoxy-7H-pyrrolo[2,3-d]pyrimidin-2-amines as potent, selective and orally bioavailable LRRK2 inhibitors
Bioorganic & Medicinal Chemistry Letters
2018
Coral: Clear and Customizable Visualization of Human Kinome Data
Cell Systems
2018
Discovery of 4-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-N-(4-((4-methylpiperazin-1-yl)methyl)phenyl)-1H-pyrazole-3-carboxamide (FN-1501), an FLT3- and CDK-Kinase Inhibitor with Potentially High Efficiency against Acute Myelocytic Leukemia
Journal of Medicinal Chemistry
2018
Targeting CDK9 Reactivates Epigenetically Silenced Genes in Cancer
Cell
2018
Kinome and phosphoproteome of high-grade meningiomas reveal AKAP12 as a central regulator of aggressiveness and its possible role in progression
Scientific Reports
2018
Discovery of N1-(4-((7-Cyclopentyl-6-(dimethylcarbamoyl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)phenyl)-N8-hydroxyoctanediamide as a Novel Inhibitor Targeting Cyclin-dependent Kinase 4/9 (CDK4/9) and Histone Deacetlyase1 (HDAC1) against Malignant Cancer
Journal of Medicinal Chemistry
2018
Discovery of Novel Potent VEGFR-2 Inhibitors Exerting Significant Antiproliferative Activity against Cancer Cell Lines
Journal of Medicinal Chemistry
2017
Development of an orally available inhibitor of CLK1 for skipping a mutated dystrophin exon in Duchenne muscular dystrophy
Scientific Reports
2017
Structural pliability adjacent to the kinase domain highlights contribution of FAK1 IDRs to cytoskeletal remodeling
Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics
2017
KinMap: a web-based tool for interactive navigation through human kinome data
BMC Bioinformatics
2017
Mapping of inhibitors and activity data to the human kinome and exploring promiscuity from a ligand and target perspective
Chemical Biology & Drug Design
2017
Phenotypic screening identifies Axl kinase as a negative regulator of an alveolar epithelial cell phenotype
Laboratory Investigation
2017
C-SPADE: a web-tool for interactive analysis and visualization of drug screening experiments through compound-specific bioactivity dendrograms
Nucleic Acids Research
2017
Annual Reports in Medicinal Chemistry
2017
Data on evolution of intrinsically disordered regions of the human kinome and contribution of FAK1 IDRs to cytoskeletal remodeling
Data in Brief
2017
Methods and Principles in Medicinal Chemistry
2017
Nuclear phosphoproteome analysis of 3T3-L1 preadipocyte differentiation reveals system-wide phosphorylation of transcriptional regulators
PROTEOMICS
2017
Potent Pan-Raf and Receptor Tyrosine Kinase Inhibitors Based on a Cyclopropyl Formamide Fragment Overcome Resistance
Journal of Chemical Information and Modeling
2017
Identifying pathogenicity of human variants via paralog-based yeast complementation
PLOS Genetics
2016
Unprecedently Large-Scale Kinase Inhibitor Set Enabling the Accurate Prediction of Compound–Kinase Activities: A Way toward Selective Promiscuity by Design?
Journal of Chemical Information and Modeling
2016
Clinical and kinomic analysis identifies peripheral blood mononuclear cells as a potential pharmacodynamic biomarker in metastatic renal cell carcinoma patients treated with sunitinib
Oncotarget
2016
Activity-Based Proteomics Reveals Heterogeneous Kinome and ATP-Binding Proteome Responses to MEK Inhibition in KRAS Mutant Lung Cancer
Proteomes
2016
Systems biological understanding of the regulatory network and the possible therapeutic strategies for vascular calcification
Molecular BioSystems
2016
Discovery and optimization of 1,7-disubstituted-2,2-dimethyl-2,3-dihydroquinazolin-4(1H)-ones as potent and selective PKCθ inhibitors
Bioorganic & Medicinal Chemistry
2016
The kinome 'at large' in cancer
Nature Reviews Cancer
2016
Integrative proteomic analysis reveals reprograming tumor necrosis factor signaling in epithelial mesenchymal transition
Journal of Proteomics
2016
Activity-Based Protein Profiling Shows Heterogeneous Signaling Adaptations to BRAF Inhibition
Journal of Proteome Research
2016
From Lead to Drug Candidate: Optimization of 3-(Phenylethynyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine Derivatives as Agents for the Treatment of Triple Negative Breast Cancer
Journal of Medicinal Chemistry
2016
AAPS Advances in the Pharmaceutical Sciences Series
2016
KLIFS: a structural kinase-ligand interaction database
Nucleic Acids Research
2015
The Nuclear Proteome of a Vertebrate
Current Biology
2015
Kovalent-allosterische Kinase-Inhibitoren
Angewandte Chemie
2015
Conformational Analysis of the DFG-Out Kinase Motif and Biochemical Profiling of Structurally Validated Type II Inhibitors
Journal of Medicinal Chemistry
2015
Covalent-Allosteric Kinase Inhibitors
Angewandte Chemie International Edition
2015
Identification of a DYRK1A Inhibitor that Induces Degradation of the Target Kinase using Co-chaperone CDC37 fused with Luciferase nanoKAZ
Scientific Reports
2015
Design and synthesis of a potent inhibitor of class 1 DYRK kinases as a suppressor of adipogenesis
Bioorganic & Medicinal Chemistry
2015
Identifying novel targets of oncogenic EGF receptor signaling in lung cancer through global phosphoproteomics
PROTEOMICS
2015
DFGmodel: Predicting Protein Kinase Structures in Inactive States for Structure-Based Discovery of Type-II Inhibitors
ACS Chemical Biology
2015
Detection of Binding Site Molecular Interaction Field Similarities
Journal of Chemical Information and Modeling
2014
Assessing adaptation of the cancer kinome in response to targeted therapies
Biochemical Society Transactions
2014
A novel small-molecule MRCK inhibitor blocks cancer cell invasion
Cell Communication and Signaling
2014
Hotspot activating PRKD1 somatic mutations in polymorphous low-grade adenocarcinomas of the salivary glands
Nature Genetics
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