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2024
Novel Drug Screening Assay for Acanthamoeba castellanii and the Anti-Amoebic Effect of Carbonic Anhydrase Inhibitors
Journal of Medicinal Chemistry
2024
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains
International Journal of Molecular Sciences
2024
Drug interactions of carbonic anhydrase inhibitors and activators
Expert Opinion on Drug Metabolism & Toxicology
2023
Synthesis, Antibacterial, and Antimonooxidase Activity of 4-(2-Methyl-1,3-oxazol-5-yl)benzenesulfonamide
Russian Journal of General Chemistry
2023
Exploring novel aryl/heteroaryl-isosteres of phenylthiazole against multidrug-resistant bacteria
RSC Advances
2023
Selected strategies to fight pathogenic bacteria
Journal of Enzyme Inhibition and Medicinal Chemistry
2023
Carbonic Anhydrase Inhibition as a Target for Antibiotic Synergy in Enterococci
Microbiology Spectrum
2023
Substituted salicylic acid analogs offer improved potency against multidrug-resistant Neisseria gonorrhoeae and good selectivity against commensal vaginal bacteria
Scientific Reports
2023
Synthesis, antibacterial and antimonooxidase activity of 4-(2-methyl-1,3-oxazol-5-yl)benzenesulfonamide
Журнал общей химии
2023
Carboxyl group-decorated polythiophenes polymeric PBTE-T-COOH for visible-light-driven photocatalytic drug-resistant bacteria inactivation
Materials Today Communications
2023
Resistance, Tolerance, Virulence and Bacterial Pathogen Fitness—Current State and Envisioned Solutions for the Near Future
Pathogens
2023
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships
Journal of Enzyme Inhibition and Medicinal Chemistry
2023
Carbonic Anhydrase Inhibitors as Novel Antibacterials in the Era of Antibiotic Resistance: Where Are We Now?
Antibiotics
2023
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates
Journal of Enzyme Inhibition and Medicinal Chemistry
2023
Evaluation of 1,3,4-Thiadiazole Carbonic Anhydrase Inhibitors for Gut Decolonization of Vancomycin-Resistant Enterococci
ACS Medicinal Chemistry Letters
2023
Antimicrobial effects of Medicines for Malaria Venture Pathogen Box compounds on strains of Neisseria gonorrhoeae
Antimicrobial Agents and Chemotherapy
2023
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ
Journal of Enzyme Inhibition and Medicinal Chemistry
2022
Repurposing FDA-approved sulphonamide carbonic anhydrase inhibitors for treatment of Neisseria gonorrhoeae
Journal of Enzyme Inhibition and Medicinal Chemistry
2022
Photocatalytic degradation of vancomycin using titanium dioxide and optimization by central composite design
International Journal of Environmental Science and Technology
2022
Mechanistic Studies and In Vivo Efficacy of an Oxadiazole-Containing Antibiotic
Journal of Medicinal Chemistry
2022
In vivo efficacy of acetazolamide in a mouse model of Neisseria gonorrhoeae infection
Microbial Pathogenesis
2022
The Use of Synchrotron Radiation in Virology
ЗДОРОВЬЕ НАСЕЛЕНИЯ И СРЕДА ОБИТАНИЯ - ЗНиСО / PUBLIC HEALTH AND LIFE ENVIRONMENT
2022
Mucoadhesive brinzolamide-loaded nanofibers for alternative glaucoma treatment
European Journal of Pharmaceutics and Biopharmaceutics
2022
Biological investigation of N-methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors
Journal of Enzyme Inhibition and Medicinal Chemistry
2021
Selective Inhibition of Helicobacter pylori Carbonic Anhydrases by Carvacrol and Thymol Could Impair Biofilm Production and the Release of Outer Membrane Vesicles
International Journal of Molecular Sciences
2021
Novel 1,3,5-Triazinyl Aminobenzenesulfonamides Incorporating Aminoalcohol, Aminochalcone and Aminostilbene Structural Motifs as Potent Anti-VRE Agents, and Carbonic Anhydrases I, II, VII, IX, and XII Inhibitors
International Journal of Molecular Sciences
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